TGR5 Receptor Agonist
TGR5 Receptor Agonist

TGR5 Receptor Agonist

Product Name: TGR5 Receptor Agonist
Synonyms: 3-(2-chlorophenyl)-N-(4-chlorophenyl)-N,5-dimethyl-4-isoxazolecarboxamideWeb Site click
Product Overview: A small molecule activator of a G protein-coupled bile acid receptor (pEC50 = 6.8-7.5) that is reported to improve GLP-1 secretion by increasing intracellular cAMP levels; used to investigate the signaling, trafficking, and regulation of TGR5 receptors in
Shipping: wet ice
CAS NO: 1538604-68-0 BLU9931
Stability: Store at -20 degrees; shelf life 730 days maximum after production
Molecular Formula: C18H14Cl2N2O2
SMILES: ClC1=C(C2=NOC(C)=C2C(N(C3=CC=C(Cl)C=C3)C)=O)C=CC=C1Natural_Product_Library_ inhibitors
Molecular Weight: 361.2
Formulation: A crystalline solid
Purity: ≥98%PubMed ID:http://www.bloodjournal.org/content/124/21/33