Product Name: OTX015
Synonyms: (6S)-4-(4-chlorophenyl)-N-(4-hydroxyphenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetamide (−)-OTX015 Medchemexpress.com
Product Overview: An orally bioavailable, small molecule inhibitor of BRD2, BRD3, and BRD4 (EC50s = 10-19 nM) that displays antiproliferative effects at a sub-micromolar range in vitro in a wide range of solid tumor types and leukemiasThe bromodomain and extra terminal dom
Shipping: wet ice
CAS NO: 6080-58-6 Product: Citric acid (trilithium salt tetrahydrate)
Stability: Store at -20 degrees; shelf life 730 days maximum after production
Molecular Formula: C25H22ClN5O2S
SMILES: ClC1=CC=C(C=C1)C2=N[[email protected]@H](CC(NC3=CC=C(O)C=C3)=O)C4=NN=C(C)N4C5=C2C(C)=C(C)S5Proton Pump inhibitors
Molecular Weight: 492
Formulation: A crystalline solid
Purity: ≥95%PubMed ID:http://aac.asm.org/content/56/6/3441.abstract