MK2 Inhibitor III
MK2 Inhibitor III

MK2 Inhibitor III

Product Name: MK2 Inhibitor III
Synonyms: 1,5,6,7-tetrahydro-2-[2-(3-quinolinyl)-4-pyridinyl]-4H-pyrrolo[3,2-c]pyridin-4-one, monohydrateWeb Site:Medchemexpress
Product Overview: A potent, cell-permeable inhibitor of MK2 (IC50 = 8.5 nM); less potently blocks MK3 and MK5 (IC50s = 210 and 81 nM, respectively) and is weak or inactive against several other kinases, including other p38 MAP kinase targets; prevents LPS-induced synthesis
Shipping: wet ice
CAS NO: 14679-73-3 Product: Todralazine
Stability: Store at -20 degrees; shelf life 730 days maximum after production
Molecular Formula: C21H16N4O • H2O
SMILES: O=C(NCC1)C2=C1NC(C3=CC(C4=CC(C=CC=C5)=C5N=C4)=NC=C3)=C2.OBradykinin Receptor inhibitors
Molecular Weight: 358.4
Formulation: A crystalline solid
Purity: ≥95%PubMed ID:http://aac.asm.org/content/56/10/5224.abstract