LGK974
LGK974

LGK974

Product Name: LGK974
Synonyms: 2,3-dimethyl-N-[5-(2-pyrazinyl)-2-pyridinyl]-[2,4-bipyridine]-5-acetamide PORCN Inhibitor IVWeb Site:Medchemexpress
Product Overview: A potent and specific small molecule inhibitor of PORCN (IC50 = 0.4 nM); greatly reduces Wnt secretion without decreasing its synthesis and without increasing cytotoxicity; orally bioavailable in micePorcupine (PORCN) is a membrane bound O-acyltransferase
Shipping: wet ice
CAS NO: 154323-57-6 Product: Almotriptan
Stability: Store at -20 degrees; shelf life 730 days maximum after production
Molecular Formula: C23H20N6O
SMILES: CC1=CC(C2=NC=C(CC(NC3=CC=C(C4=CN=CC=N4)C=N3)=O)C=C2C)=CC=N1GNRH Receptor inhibitors
Molecular Weight: 396.4
Formulation: A crystalline solid
Purity: ≥98%PubMed ID:http://aac.asm.org/content/57/1/83.abstract