GSK1016790A
GSK1016790A

GSK1016790A

Product Name: GSK1016790A
Synonyms: N-[(1S)-1-[[4-[(2S)-2-[[(2,4-dichlorophenyl)sulfonyl]amino]-3-hydroxy-1-oxopropyl]-1-piperazinyl]carbonyl]-3-methylbutyl]-benzo[b]thiophene-2-carboxamideMedchemexpress
Product Overview: A TRPV4 agonist that has been reported to elicit calcium influx in HEK cells expressing mouse or human TRPV4 (EC50s = 18 and 2.1 nM, respectively); used to demonstrate a role for TRPV4 in regulating urinary bladder activity and endothelial control of vasc
Shipping: wet ice
CAS NO: 208255-80-5 DAPT
Stability: Store at -20 degrees; shelf life 730 days maximum after production
Molecular Formula: C28H32Cl2N4O6S2
SMILES: ClC1=CC=C(S(N[[email protected]](C(N2CCN(C([[email protected]@H](NC(C3=CC4=C(C=CC=C4)S3)=O)CC(C)C)=O)CC2)=O)CO)(=O)=O)C(Cl)=C1Neuropeptide Y Receptor inhibitors
Molecular Weight: 655.6
Formulation: A crystalline solid
Purity: ≥98%PubMed ID:http://www.bloodjournal.org/content/129/1/128