Darapladib
Darapladib

Darapladib

Product Name: Darapladib
Synonyms: N-[2-(diethylamino)ethyl]-2-[[(4-fluorophenyl)methyl]thio]-4,5,6,7-tetrahydro-4-oxo-N-[[4-(trifluoromethyl)[1,1-biphenyl]-4-yl]methyl]-1H-cyclopentapyrimidine-1-acetamide Medchemexpress.com
Product Overview: A reversible inhibitor of Lp-PLA2 (IC50 = 0.25 nM) that produces sustained inhibition of plasma Lp-PLA2 activity in humansLipoprotein-associated phospholipase A2 (Lp-PLA2), also known as platelet activating factor acetylhydrolase (PAF-AH) or phospholipase
Shipping: wet ice
CAS NO: 166095-21-2 Product: BMS-191095
Stability: Store at -20 degrees; shelf life 730 days maximum after production
Molecular Formula: C36H38F4N4O2S
SMILES: FC1=CC=C(CSC2=NC(C(CCC3)=C3N2CC(N(CC4=CC=C(C5=CC=C(C(F)(F)F)C=C5)C=C4)CCN(CC)CC)=O)=O)C=C1BMX Kinase inhibitors
Molecular Weight: 666.8
Formulation: A crystalline solid
Purity: ≥98%PubMed ID:http://aac.asm.org/content/55/10/4594.abstract