Product Name: CPI-360
Synonyms: N-[(1,2-dihydro-4-methoxy-6-methyl-2-oxo-3-pyridinyl)methyl]-2-methyl-1-[(1R)-1-(tetrahydro-2H-pyran-4-yl)ethyl]-1H-indole-3-carboxamideMedchemexpress.com
Product Overview: A selective EZH2 inhibitor (IC50s = 0.5 and 2.5 nM for wild-type EZH2 and Y641N mutant EZH2, respectively); decreases cellular levels of H3K27me3 and H3K27me2 (EC50s = 56 and 65 nM, respectively), triggering cell cycle arrest and ultimately resulting in a
Shipping: wet ice
CAS NO: 35943-35-2 Product: Triciribine
Stability: Store at -20 degrees; shelf life 730 days maximum after production
Molecular Formula: C25H31N3O4
SMILES: CC(N1)=CC(OC)=C(CNC(C2=C(C)N([C@H](C)C3CCOCC3)C4=C2C=CC=C4)=O)C1=OMelatonin Receptor inhibitors
Molecular Weight: 437.5
Formulation: A crystalline solid
Purity: ≥98%PubMed ID:http://aac.asm.org/content/60/4/2528.abstract
