BX-795
BX-795

BX-795

Product Name: BX-795
Synonyms: N-[3-[[5-iodo-4-[[3-[(2-thienylcarbonyl)amino]propyl]amino]-2-pyrimidinyl]amino]phenyl]-1-pyrrolidinecarboxamideWeb Site click
Product Overview: A potent, ATP-competitive inhibitor of PDK1 in vitro (IC50 = 11 nM) and in cells (IC50 = 300 nM); also inhibits ERK8, MNK2, Aurora B, Aurora C, MARKs 1-4,TBK1, IKKε, and additional kinases at comparable concentrations3-Phosphoinositide-dependent p
Shipping: wet ice
CAS NO: Product: Prochlorperazine (D8 dimeleate)
Stability: Store at -20 degrees; shelf life 730 days maximum after production
Molecular Formula: C23H26IN7O2S
SMILES: [H]N(CCCN(C(C1=CC=CS1)=O)[H])C2=C(I)C=NC(N([H])C3=CC(N(C(N4CCCC4)=O)[H])=CC=C3)=N2GPR109A inhibitors
Molecular Weight: 591.5
Formulation: A crystalline solid
Purity: ≥98%PubMed ID:http://aac.asm.org/content/56/1/352.abstract