Product Name: RQ-00203078
Synonyms: 4-[[[3-chloro-5-(trifluoromethyl)-2-pyridinyl][[4-(trifluoromethoxy)phenyl]methyl]amino]sulfonyl]-benzoic acidMedchemexpress
Product Overview: A selective TRPM8 antagonist (IC50s = 8.3 and 5.8 nM in human and rat, respectively); attenuates icilin-induced wet-dog shakes in rats (ED50 = 0.65 mg/kg); reduces HSC3 and HSC4 oral squamous carcinoma cell migration and invasion in vitroRQ-00203078 is a
Shipping: wet ice
CAS NO: 869901-69-9 Product: MK-2048
Stability: Store at -20 degrees; shelf life 730 days maximum after production
Molecular Formula: C21H13ClF6N2O5S
SMILES: OC(C1=CC=C(S(N(CC2=CC=C(OC(F)(F)F)C=C2)C3=NC=C(C(F)(F)F)C=C3Cl)(=O)=O)C=C1)=OPARP inhibitors
Molecular Weight: 554.8
Formulation: A crystalline solid
Purity: ≥98%PubMed ID:http://aac.asm.org/content/60/3/1289.abstract
