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Product Name: PFI-1
Synonyms: 2-methoxy-N-(3-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-6-yl)benzenesulfonamide PF-06405761Web Site:Medchemexpress
Product Overview: A BET bromodomain inhibitor that exhibits inhibitory activity at BRD2 bromodomain 2 and BRD4 bromodomain 1 with IC50 values of 98 nM and 0.22 μM, respectivelyBromodomains recognize acetylated lysine residues and recruit regulatory complexes to acetylat
Shipping: wet ice
CAS NO: 300816-15-3 RS 504393
Stability: Store at -20 degrees; shelf life 730 days maximum after production
Molecular Formula: C16H17N3O4S
SMILES: O=S(C1=C(OC)C=CC=C1)(NC2=CC=C(NC(N(C)C3)=O)C3=C2)=ODeubiquitinase inhibitors
Molecular Weight: 347.4
Formulation: A crystalline solid
Purity: ≥98%PubMed ID:http://www.bloodjournal.org/content/129/21/2857

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Author: signsin1dayinc