ICI 216140

Product Name: ICI 216140
Synonyms: N-(2-methyl-1-oxopropyl)-7-D-alanine-9-(N-methyl-L-leucinamide)-3-9-neuromedin CWeb Site:Medchemexpress
Product Overview: A GRP/bombesin receptor 2 antagonist (IC50 = 4.13 nM in vitro); reduces bombesin-stimulated pancreatic amylase secretion and attenuates bombesin-stimulated increases in blood pressure in ratsBombesin is a peptide, originally isolated from the skin of the
Shipping: wet ice
CAS NO: 60940-34-3 Ebselen
Stability: Store at -20 degrees; shelf life 730 days maximum after production
Molecular Formula: C45H65N13O8
SMILES: CC(C)C(N[[email protected]@H](CC1=CNC=N1)C(N[[email protected]@H](CC2=CNC3=C2C=CC=C3)C(N[[email protected]@H](C)C(N[[email protected]@H](C(C)C)C(N[[email protected]](C)C(N[[email protected]@H](CC4=CNC=N4)C(N[[email protected]@H](CC(C)C)C(NC)=O)=O)=O)=O)=O)=O)=O)=OGlucokinase inhibitors
Molecular Weight: 916.1
Formulation: A crystalline solid
Purity: ≥95%PubMed ID:http://www.bloodjournal.org/content/127/4/392