Product Name: I-BET151
Synonyms: 7,3,5-dimethyl-4-isoxazolyl-1,3-dihydro-8-methoxy-1-[1R-1-(2-pyridinyl)ethyl]-2H-imidazo[4,5-c]quinolin-2-one GSK1210151AWeb Site：Medchemexpress
Product Overview: An isoxazole class pan-BET family inhibitor, blocking BRD2, BRD3, and BRD4 with IC50 values of 0.5, 0.25, and 0.79 µM, respectively); induces apoptosis or triggers G0/G1 cell cycle arrest in MLL-fusion cell lines; effective in vivo, suppressing MLL
Shipping: wet ice
CAS NO: 127-58-2 Product: Sulfamerazine (sodium salt)
Stability: Store at -20 degrees; shelf life 730 days maximum after production
Molecular Formula: C23H21N5O3
SMILES: CC(ON=C1C)=C1C2=CC(N=CC(N3)=C4N([C@H](C)C5=CC=CC=N5)C3=O)=C4C=C2OCCXCR inhibitors
Molecular Weight: 415.5
Formulation: A crystalline solid
Purity: ≥98%PubMed ID:http://aac.asm.org/content/58/8/4902.abstract
