Product Name: GSK2830371
Synonyms: 5-[[(5-chloro-2-methyl-3-pyridinyl)amino]methyl]-N-[(1S)-1-(cyclopentylmethyl)-2-(cyclopropylamino)-2-oxoethyl]-2-thiophenecarboxamideMedchemexpress.com
Product Overview: A potent and selective inhibitor of Wip1 (IC50 = 6 nM); increases phosphorylation of Wip1 substrates and blocks cell cycling in cancer cells; orally bioavailable, causing inhibition of lymphoma xenograft growth in miceThe wild-type p53-induced phosphatase
Shipping: wet ice
CAS NO: 1332708-14-1 PF-4840154
Stability: Store at -20 degrees; shelf life 730 days maximum after production
Molecular Formula: C23H29ClN4O2S
SMILES: ClC1=CC(NCC2=CC=C(C(N[C@H](C(NC3CC3)=O)CC4CCCC4)=O)S2)=C(C)N=C1ATP Synthase inhibitors
Molecular Weight: 461
Formulation: A crystalline solid
Purity: ≥98%PubMed ID:http://www.bloodjournal.org/content/129/15/2132
