Product Name: EPZ011989
Synonyms: N-[(1,2-dihydro-4,6-dimethyl-2-oxo-3-pyridinyl)methyl]-3-[ethyl[trans-4-[(2-methoxyethyl)methylamino]cyclohexyl]amino]-2-methyl-5-[3-(4-morpholinyl)-1-propyn-1-yl]-benzamideMedchemexpress
Product Overview: A selective, orally bioavailable EZH2 inhibitor with Ki values that are less than 3 nM for wild type and Tyr646 mutant of EZH2; demonstrates significant tumor growth inhibition in a mouse xenograft model of human B cell lymphomaThe lysine methyltransferas
Shipping: wet ice
CAS NO: 1029712-80-8 Product: INCB28060
Stability: Store at -20 degrees; shelf life 730 days maximum after production
Molecular Formula: C35H51N5O4
SMILES: CN(CCOC)[C@@H]1CC[C@@H](N(C2=CC(C#CCN3CCOCC3)=CC(C(NCC4=C(C)C=C(C)NC4=O)=O)=C2C)CC)CC1Anti-cancer_Compound_Library inhibitors
Molecular Weight: 605.8
Formulation: A crystalline solid
Purity: ≥98%PubMed ID:http://aac.asm.org/content/59/10/5992.abstract
