Product Name: EI1
Synonyms: 6-cyano-N-[(1,2-dihydro-4,6-dimethyl-2-oxo-3-pyridinyl)methyl]-1-(1-ethylpropyl)-1H-indole-4-carboxamideMedchemexpress.com
Product Overview: A selective EZH2 inhibitor that has activity against both wild-type and Y641F mutant EZH2 (IC50s = 15 and 13 nM, respectively); blocks cellular H3K27 methylation and activates PRC2-specific gene expression; decreases proliferation, cell cycle arrest, and
Shipping: wet ice
CAS NO: 380315-80-0 Product: Tenovin-1
Stability: Store at -20 degrees; shelf life 730 days maximum after production
Molecular Formula: C23H26N4O2
SMILES: O=C(NCC1=C(C)C=C(C)NC1=O)C2=CC(C#N)=CC3=C2C=CN3C(CC)CCPhosphatase_Inhibitor_Cocktail_II inhibitors
Molecular Weight: 390.5
Formulation: A crystalline solid
Purity: ≥98%PubMed ID:http://aac.asm.org/content/59/10/5967.abstract
