Product Name: BMS 754807
Synonyms: 1-[4-[(5-cyclopropyl-1H-pyrazol-3-yl)amino]pyrrolo[2,1-f][1,2,4]triazin-2-yl]-N-(6-fluoro-3-pyridinyl)-2-methyl-(2S)-2-pyrrolidinecarboxamideMedchemexpress
Product Overview: A reversible, orally bioavailable dual inhibitor of IGF-1R and InsR tyrosine kinases (IC50s = 1.8 and 1.7 nM, respectively); inhibits cell proliferation or induces apoptosis in a variety of cancer cells in vitro; inhibits the growth of tumor xenografts in
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CAS NO: 905854-02-6 Tivantinib
Stability: Store at -20 degrees; shelf life 730 days maximum after production
Molecular Formula: C23H24FN9O
SMILES: FC1=NC=C(NC([C@]2(C)CCCN2C3=NN4C(C(NC5=NNC(C6CC6)=C5)=N3)=CC=C4)=O)C=C1Telomerase inhibitors
Molecular Weight: 461.5
Formulation: A crystalline solid
Purity: ≥98%PubMed ID:http://www.bloodjournal.org/content/129/20/2819
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Product Name: BMS-754807
Synonyms: Web Site click
Product Overview: BMS-754807 is a potent and reversible inhibitor of IGF-1R/InsR with IC50 of 1.8 nM/1.7 nM in cell-free assays, less potent to Met, Aurora A/B, TrkA/B and Ron, and shows little activity to Flt3, Lck, MK2, PKA, PKC etc. Phase 2.
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CAS NO: 74578-69-1 Product: Ceftriaxone (sodium salt)
Stability: Store at +4 degrees; shelf life 730 days maximum after production
Molecular Formula: C23H24FN9O
SMILES: KLF inhibitors
Molecular Weight: 461.49
Formulation: solution 10mM in DMSO
Purity: 0.98PubMed ID:http://aac.asm.org/content/46/10/3276.abstract