Product Name: BIX 02565
Synonyms: (5R)-N-[1-[3-(dimethylamino)propyl]-1H-benzimidazol-2-yl]-2,3,4,5-tetrahydro-5-methyl-1-oxo-1H-[1,4]diazepino[1,2-a]indole-8-carboxamideMedchemexpress
Product Overview: A potent RSK2 inhibitor (IC50 = 1.1 nM) that also demonstrates off-target binding at multiple adrenergic receptor subtypes that are important for vascular tone and cardiac function (IC50s = 0.052-1.820 μM for adrenergic α1A, α1B, α1D,
Shipping: wet ice
CAS NO: 1072959-67-1 Product: SR-3677
Stability: Store at -20 degrees; shelf life 730 days maximum after production
Molecular Formula: C26H30N6O2
SMILES: O=C1C(N2[C@H](C)CCN1)=CC3=C2C=C(C(NC4=NC(C=CC=C5)=C5N4CCCN(C)C)=O)C=C3STAT inhibitors
Molecular Weight: 458.6
Formulation: A crystalline solid
Purity: ≥98%PubMed ID:http://aac.asm.org/content/59/8/5022.abstract
