Product Name: ARN-509
Synonyms: 4-[7-[6-cyano-5-(trifluoromethyl)-3-pyridinyl]-8-oxo-6-thioxo-5,7-diazaspiro[3.4]oct-5-yl]-2-fluoro-N-methyl-benzamide JNJ-56021927Web Site：Medchemexpress
Product Overview: An orally bioavailable antagonist of the androgen receptor (IC50 = 16 nM); at 30 mg/kg/d, suppresses tumor growth in a mouse model of castration-resistant prostate cancerARN-509 is an antagonist of the androgen receptor (IC50 = 16 nM). It binds the recep
Shipping: wet ice
CAS NO: 1337531-36-8 GSK2606414
Stability: Store at -20 degrees; shelf life 730 days maximum after production
Molecular Formula: C21H15F4N5O2S
SMILES: S=C(N(C1=CC(F)=C(C(NC)=O)C=C1)C2(CCC2)C3=O)N3C4=CN=C(C#N)C(C(F)(F)F)=C4Gap Junction Protein inhibitors
Molecular Weight: 477.4
Formulation: A crystalline solid
Purity: ≥98%PubMed ID:http://aac.asm.org/content/54/2/940.abstract
